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Cayman Brd4770; Purity- Greater Than Or Equal To 98%; Size- 1 Mg
Cayman Brd4770; Purity- Greater Than Or Equal To 98%; Size- 1 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$32.00
Your Price
$32.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-11787-1 |
MFG.PART: | 11787-1 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
BRD4770 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, decreasing di- and trimethylation on lysine 9 of histone 3 (EC50 = 5 µM). Through its effects on EHMT2, BRD4770 induces senescence in the pancreatic cancer cell line PANC-1 without initiating apoptosis. It also blocks both anchorage-
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
2- (benzoylamino)- 1- (3- phenylpropyl)- 1H- benzimidazole- 5- carboxylic acid, methyl ester
CAS Number
1374601-40-7
Synonyms
- HMTase Inhibitor VI
Molecular Formula
C25H23N3O3
Formula Weight
413.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 20 mg/ml
- DMF:PBS(pH7.2) (1:2): 0.25 mg/ml
- DMSO: 10 mg/ml
λmax
232, 271, 329 nm
SMILES
O=C(C1=CC=CC=C1)NC2=NC3=CC(C(OC)=O)=CC=C3N2CCCC4=CC=CC=C4
InChi Code
InChI=1S/C25H23N3O3/c1-31-24(30)20-14-15-22-21(17-20)26-25(27-23(29)19-12-6-3-7-13-19)28(22)16-8-11-18-9-4-2-5-10-18/h2-7,9-10,12-15,17H,8,11,16H2,1H3,(H,26,27,29)
InChi Key
UCGWYCMPZXDHNR-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-11787-1 |
---|---|
Supplier Part Number | 11787-1 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer Name | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/11787m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | CN |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 1374601-40-7 |