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Cayman Abt-869; Purity- Greater Than Or Equal To 98%; Size- 5 Mg
Cayman Abt-869; Purity- Greater Than Or Equal To 98%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$99.00
Your Price
$99.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-13653-5 |
MFG.PART: | 13653-5 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
Tolvaptan is a nonpeptide vasopressin V2 receptor antagonist (IC50 = 3 nM for rat receptor) and a diuretic agent. It is selective for V2 over V1 receptors (IC50 = 0.58 μM). Tolvaptan increases urine volume by 3-fold in rats when administered at a dose of 0.54 mg/kg. It also reduces left ventricular end-systolic volumes and improves left ventricular ejection fraction in a rat model of myocardial infarction. Formulations containing tolvaptan have been used to treat hyponatremia.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[4-[(7- chloro- 2,3,4,5- tetrahydro- 5-hydroxy- 1H-1- benzazepin-1-yl) carbonyl]-3- methylphenyl]- 2-methyl- benzamide
CAS Number
150683-30-0
Synonyms
- OPC 41061
Molecular Formula
C26H25ClN2O3
Formula Weight
448.9
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
- DMSO:PBS(pH 7.2) (1:3): 0.25 mg/mL
- Ethanol: 12 mg/mL
λmax
269 nm
SMILES
CC1=C(C(NC2=CC(C)=C(C(N3C(C=CC(Cl)=C4)=C4C(O)CCC3)=O)C=C2)=O)C=CC=C1
InChi Code
InChI=1S/C26H25ClN2O3/c1-16-6-3-4-7-20(16)25(31)28-19-10-11-21(17(2)14-19)26(32)29-13-5-8-24(30)22-15-18(27)9-12-23(22)29/h3-4,6-7,9-12,14-15,24,30H,5,8,13H2,1-2H3,(H,28,31)
InChi Key
GYHCTFXIZSNGJT-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-13653-5 |
---|---|
Supplier Part Number | 13653-5 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer Name | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/13653m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 5 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | Y |
CAS Number | 796967-16-3 |